SCHEMBL24671298

SCHEMBL24671298

O=C(Nc1ccc(C2=CCNCC2)c(F)c1)c1ccc(C2=CCNCC2)s1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ESRRG P62508 12/20 0.43
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
PTPN2 P17706 1/20 0.39
PTPN11 Q06124 1/20 0.39
HTR6 P50406 1/20 0.39
CCNT1 O60563 1/20 0.38
CDK9 P50750 1/20 0.38
ESR1 P03372 3/20 0.38
ESR2 Q92731 3/20 0.38
KDM4E B2RXH2 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
MAPKAPK2 P49137 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29803840 0.94 MAPT (0.39) ESRRGTP53MAPTHTR6ESR1
SCHEMBL24671263 0.87 KDM4E (0.42) ESRRGTP53MAPTESR1ESR2
SCHEMBL24669946 0.85 TP53 (0.42) ESRRGTP53HTR6CCNT1CDK9
SCHEMBL24670406 0.85 IMPDH2 (0.45) CCNT1CDK9KDM4EMAPKAPK2
Trifluoroacetic Acid SCHEMBL29803663 0.83 KDM4E (0.40) ESRRGTP53MAPTHTR6ESR1
SCHEMBL29803733 0.83 MAPKAPK2 (0.52) ESRRGTP53MAPTPTPN2PTPN11
SCHEMBL24670483 0.82 ULK1 (0.41) MAPTHTR6CCNT1CDK9MAPKAPK2
SCHEMBL29804024 0.82 CCNT1 (0.51) HTR6CCNT1CDK9MAPKAPK2
Trifluoroacetic Acid SCHEMBL29803398 0.81 IMPDH2 (0.41) CCNT1CDK9KDM4E
Trifluoroacetic Acid SCHEMBL29803752 0.80 WDR5 (0.41) ESRRGTP53MAPTHTR6CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed