SCHEMBL24671269

SCHEMBL24671269

CC(C)(C)OC(=O)N1CC=C(c2ccc(C(=O)Nc3ccc4c(c3)CN(C(=O)OC(C)(C)C)CC4)cc2)CC1

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 5/20 0.63
NR1H2 P55055 1/20 0.53
TMPRSS2 O15393 4/20 0.49
ESR2 Q92731 1/20 0.48
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
PIK3CA P42336 1/20 0.47
MTOR P42345 1/20 0.47
SCN9A Q15858 1/20 0.44
CDK7 P50613 1/20 0.44
CDK13 Q14004 1/20 0.44
CDK12 Q9NYV4 1/20 0.44
GRAMD1A Q96CP6 1/20 0.44
WNT3A P56704 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29803436 1.00 NAMPT (0.63) NAMPTNR1H2TMPRSS2ESR2NPC1
SCHEMBL24670854 0.95 NAMPT (0.67) NAMPTNR1H2TMPRSS2ESR2NPC1
SCHEMBL29803636 0.95 NAMPT (0.67) NAMPTNR1H2TMPRSS2ESR2NPC1
SCHEMBL30182726 0.94 NAMPT (0.68) NAMPTTMPRSS2PIK3CAMTOR
SCHEMBL24892302 0.94 NAMPT (0.68) NAMPTTMPRSS2PIK3CAMTOR
SCHEMBL29803570 0.90 NAMPT (0.58) NAMPTNR1H2TMPRSS2ESR2NPC1
SCHEMBL24670163 0.88 NAMPT (0.51) NAMPTNR1H2TMPRSS2ESR2NPC1
SCHEMBL29803391 0.88 NAMPT (0.51) NAMPTNR1H2TMPRSS2ESR2NPC1
SCHEMBL24670154 0.87 NAMPT (0.52) NAMPTNR1H2TMPRSS2ESR2NPC1
SCHEMBL24669379 0.87 NR1H2 (0.49) NAMPTNR1H2TMPRSS2ESR2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed