SCHEMBL24671434

SCHEMBL24671434

Cc1cc(C2=CCN(C(=O)OC(C)(C)C)CC2)ccc1C(=O)Nc1ccc2c(c1)CCN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 11/20 0.61
ESR2 Q92731 1/20 0.49
TMPRSS2 O15393 2/20 0.46
NR1H2 P55055 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
WNT3A P56704 1/20 0.43
PRMT5 O14744 2/20 0.42
WDR77 Q9BQA1 2/20 0.42
PIK3CA P42336 1/20 0.42
MTOR P42345 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29803581 1.00 NAMPT (0.61) NAMPTESR2TMPRSS2NR1H2NPC1
SCHEMBL29803570 0.97 NAMPT (0.58) NAMPTESR2TMPRSS2NR1H2NPC1
SCHEMBL29803727 0.96 NAMPT (0.61) NAMPTESR2TMPRSS2NR1H2NPC1
SCHEMBL24671281 0.96 NAMPT (0.61) NAMPTESR2TMPRSS2NR1H2NPC1
SCHEMBL29803738 0.87 NAMPT (0.54) NAMPTWNT3APRMT5WDR77
SCHEMBL24671269 0.87 NAMPT (0.63) NAMPTESR2TMPRSS2NR1H2NPC1
SCHEMBL29803436 0.87 NAMPT (0.63) NAMPTESR2TMPRSS2NR1H2NPC1
SCHEMBL24670854 0.86 NAMPT (0.67) NAMPTESR2TMPRSS2NR1H2NPC1
SCHEMBL29803636 0.86 NAMPT (0.67) NAMPTESR2TMPRSS2NR1H2NPC1
SCHEMBL24892052 0.85 NAMPT (0.61) NAMPTWNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed