SCHEMBL24671581

SCHEMBL24671581

COc1cc(NC(=O)c2ccc(C3=CCN(C(=O)OC(C)(C)C)CC3)c(F)c2)ncc1C1=CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 1/20 0.45
SCN9A Q15858 1/20 0.44
CDK9 P50750 4/20 0.44
GRM5 P41594 6/20 0.44
GRM1 Q13255 6/20 0.44
PDK4 Q16654 1/20 0.42
NAMPT P43490 1/20 0.42
CCNT1 O60563 2/20 0.42
EED O75530 1/20 0.41
RBBP4 Q09028 1/20 0.41
SUZ12 Q15022 1/20 0.41
EZH2 Q15910 1/20 0.41
FGFR1 P11362 1/20 0.41
DGAT2 Q96PD7 1/20 0.41
GPR119 Q8TDV5 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24671483 0.93 JAK1 (0.42) JAK1SCN9ACDK9GRM5GRM1
SCHEMBL24671417 0.87 GRM1 (0.47) JAK1SCN9ACDK9GRM5GRM1
SCHEMBL29803582 0.87 GRM1 (0.47) JAK1SCN9ACDK9GRM5GRM1
SCHEMBL29803476 0.87 NAMPT (0.49) JAK1SCN9ACDK9GRM5GRM1
SCHEMBL24670963 0.86 CCNT1 (0.40) CDK9CCNT1
SCHEMBL29803589 0.86 CDK9 (0.37) JAK1SCN9ACDK9CCNT1EED
SCHEMBL24670970 0.86 CDK9 (0.37) JAK1SCN9ACDK9CCNT1EED
SCHEMBL24670962 0.86 CDK9 (0.37) JAK1SCN9ACDK9CCNT1EED
SCHEMBL24669383 0.86 NAMPT (0.49) JAK1SCN9ACDK9GRM5GRM1
SCHEMBL29803406 0.86 NAMPT (0.49) JAK1SCN9ACDK9GRM5GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed