SCHEMBL24671483

SCHEMBL24671483

COc1cc(NC(=O)c2ccc(C3=CCNCC3)c(F)c2)ncc1C1=CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 1/20 0.42
CDK9 P50750 7/20 0.41
CCNT1 O60563 5/20 0.40
SCN9A Q15858 1/20 0.40
EED O75530 1/20 0.39
RBBP4 Q09028 1/20 0.39
SUZ12 Q15022 1/20 0.39
EZH2 Q15910 1/20 0.39
GRM5 P41594 4/20 0.39
GRM1 Q13255 4/20 0.39
TNF P01375 1/20 0.38
PDK4 Q16654 1/20 0.38
NAMPT P43490 1/20 0.38
WDR5 P61964 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24671581 0.93 JAK1 (0.45) JAK1CDK9CCNT1SCN9AEED
SCHEMBL29803778 0.87 CCNT1 (0.50) CDK9CCNT1
SCHEMBL24671479 0.87 CCNT1 (0.50) CDK9CCNT1
SCHEMBL24671033 0.86 GRM1 (0.44) JAK1CDK9CCNT1SCN9AGRM5
SCHEMBL24671474 0.81 WNT3A (0.45) CDK9CCNT1NAMPT
SCHEMBL29803476 0.81 NAMPT (0.49) JAK1CDK9CCNT1SCN9AGRM5
SCHEMBL29803582 0.81 GRM1 (0.47) JAK1CDK9CCNT1SCN9AEED
SCHEMBL24671417 0.81 GRM1 (0.47) JAK1CDK9CCNT1SCN9AEED
SCHEMBL24670963 0.81 CCNT1 (0.40) CDK9CCNT1
SCHEMBL24670962 0.81 CDK9 (0.37) JAK1CDK9CCNT1SCN9AEED

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed