SCHEMBL24672012

SCHEMBL24672012

C=Cc1c(N)nc(C)nc1Cl

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
MAPK1 P28482 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29698777 0.78 LMNA (0.40) HTTSMN1; SMN2KDM4ELMNANPSR1
SCHEMBL24096383 0.78 LMNA (0.40) HTTSMN1; SMN2KDM4ELMNANPSR1
SCHEMBL24671926 0.75 LRRK2 (0.31)
SCHEMBL115474 0.73 HTT (0.33) HTTSMN1; SMN2ALDH1A1
SCHEMBL8532660 0.72 KDM4E (0.39) HTTSMN1; SMN2KDM4ELMNAMAPK1
SCHEMBL16461044 0.72 LMNA (0.40) SMN1; SMN2KDM4ELMNA
SCHEMBL14165804 0.72 HTT (0.35) HTTSMN1; SMN2LMNAALDH1A1
SCHEMBL259072 0.72 PDE10A (0.52) HTTSMN1; SMN2LMNAALDH1A1
SCHEMBL29484711 0.72 HTT (0.35) HTTSMN1; SMN2LMNAALDH1A1
SCHEMBL116212 0.72 HTT (0.37) HTTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116669738-A Pyrimidopyridone derivative as SOS1 inhibitor, and preparation method and application thereof 苏州阿尔脉生物科技有限公司 2023-08-29 CN disclosed
WO-2022170802-A1 PYRIMIDO-PYRIDONE DERIVATIVE AS SOS1 INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF 苏州阿尔脉生物科技有限公司 2022-08-18 WO disclosed
WO-2022170802-A1 PYRIMIDO-PYRIDONE DERIVATIVE AS SOS1 INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF 苏州阿尔脉生物科技有限公司 2022-08-18 WO disclosed