SCHEMBL24676049

SCHEMBL24676049

CC(C)(C)[Si](C)(C)OC1CCC(c2nc(C(F)(F)F)cs2)C1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 3/20 0.39
HCRTR2 O43614 2/20 0.31
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31
APH1B Q8WW43 1/20 0.31
NCSTN Q92542 1/20 0.31
APH1A Q96BI3 1/20 0.31
PSENEN Q9NZ42 1/20 0.31
HCRTR1 O43613 1/20 0.31
SPR P35270 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24676040 0.91 TRPV1 (0.34) TRPV1PSEN1PSEN2APH1BNCSTN
SCHEMBL24676509 0.91 TRPV1 (0.34) TRPV1PSEN1PSEN2APH1BNCSTN
SCHEMBL25164697 0.76 TRPV1 (0.41) TRPV1HCRTR2PSEN1PSEN2APH1B
SCHEMBL29754965 0.76 TRPV1 (0.37) TRPV1HCRTR2PSEN1PSEN2APH1B
SCHEMBL24676720 0.75
SCHEMBL24676986 0.74 CHRM2 (0.33)
SCHEMBL29754833 0.73
SCHEMBL24676724 0.73 OGA (0.34) TRPV1
SCHEMBL29754880 0.73 TRPV1 (0.43) TRPV1HCRTR2PSEN1PSEN2APH1B
SCHEMBL29754886 0.73 TRPV1 (0.43) TRPV1HCRTR2PSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed