SCHEMBL24676469

SCHEMBL24676469

CN(C(=O)OC(C)(C)C)c1nc(C(F)(F)F)c(-c2ccnc(Cl)n2)s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 6/20 0.39
PAX8 Q06710 1/20 0.37
ATF1 P18846 2/20 0.35
NFKB1 P19838 2/20 0.35
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
CDK1 P06493 3/20 0.33
CCNB1 P14635 3/20 0.33
CCNA2 P20248 3/20 0.33
CDK2 P24941 3/20 0.33
CDK7 P50613 3/20 0.33
CCNH P51946 3/20 0.33
CCNT1 O60563 2/20 0.33
CDK9 P50750 2/20 0.33
CCNA1 P78396 2/20 0.33
CDK4 P11802 1/20 0.31
CCND1 P24385 1/20 0.31
CCND3 P30281 1/20 0.31
CDK6 Q00534 1/20 0.31
GABRA1 P14867 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29754868 0.75 PAX8 (0.37) PAX8ALOX15TSHRABL1USP30
SCHEMBL24676942 0.75 CDK2 (0.43) CDK1CCNB1CCNA2CDK2CDK7
SCHEMBL24676941 0.75 IKBKB (0.48) CDK1CCNB1CCNA2CDK2CDK7
SCHEMBL28509124 0.74 CDK2 (0.51) AAK1PAX8ALOX15TSHRCDK2
SCHEMBL8083910 0.74 PAX8 (0.52) AAK1PAX8SYK
SCHEMBL448042 0.72 SYK (0.38) AAK1PAX8SYKSSTR4USP30
SCHEMBL24676006 0.72 GPBAR1 (0.34) PAX8ATF1NFKB1ABL1GPBAR1
SCHEMBL29755073 0.72 GPBAR1 (0.34) PAX8ATF1NFKB1ABL1GPBAR1
SCHEMBL24676013 0.70 PAX8 (0.33) AAK1PAX8ATF1NFKB1SYK
SCHEMBL30926187 0.70 STK17B (0.36) PAX8ALOX15TSHRCDK1SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed