SCHEMBL24676597

SCHEMBL24676597

CN(C)Cc1nc(C(F)(F)F)c(-c2nc(NC3CCNCC3)ncc2F)s1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 13/20 0.37
CDK9 P50750 11/20 0.37
CCNT1 O60563 10/20 0.37
CDK4 P11802 8/20 0.37
CCND1 P24385 8/20 0.37
CDK7 P50613 7/20 0.37
CCNA2 P20248 7/20 0.37
CCND3 P30281 7/20 0.37
CDK6 Q00534 7/20 0.37
CCNH P51946 6/20 0.37
CDK1 P06493 4/20 0.37
CCNB1 P14635 4/20 0.37
PTK2 Q05397 1/20 0.37
CCNK O75909 6/20 0.35
CDK12 Q9NYV4 6/20 0.35
CCNE1 P24864 6/20 0.35
CSNK1A1 P48729 1/20 0.34
CDK13 Q14004 1/20 0.34
MNAT1 P51948 1/20 0.34
MAPK8 P45983 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29754815 1.00 CDK2 (0.37) CDK2CDK9CCNT1CDK4CCND1
SCHEMBL24676943 0.89 CDK9 (0.33) CDK2CDK9CCNT1CDK4CCND1
SCHEMBL29754894 0.89 CDK9 (0.33) CDK2CDK9CCNT1CDK4CCND1
SCHEMBL24676684 0.85 CDK2 (0.43) CDK2CDK9CCNT1CDK4CCND1
SCHEMBL24676566 0.84 CCNE1 (0.45) CDK2CDK9CCNT1CDK4CCND1
SCHEMBL29754806 0.84 CDK2 (0.54) CDK2CDK4CCND1CCNA2CCND3
SCHEMBL24676105 0.84 CDK2 (0.36) CDK2CDK9CCNT1CDK4CCND1
SCHEMBL24676765 0.84 CDK2 (0.54) CDK2CDK4CCND1CCNA2CCND3
SCHEMBL24676764 0.84 CDK2 (0.36) CDK2CDK9CCNT1CDK4CCND1
SCHEMBL24676103 0.83 CCNE1 (0.47) CDK2CDK9CCNT1CDK4CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed