SCHEMBL24676943

SCHEMBL24676943

CC1CC(Nc2ncc(F)c(-c3sc(CN(C)C)nc3C(F)(F)F)n2)CCN1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 8/20 0.33
CDK7 P50613 6/20 0.33
CCNK O75909 4/20 0.33
CDK12 Q9NYV4 4/20 0.33
CSNK1A1 P48729 1/20 0.33
CDK13 Q14004 1/20 0.33
CDK2 P24941 9/20 0.32
CCNT1 O60563 7/20 0.32
CDK4 P11802 6/20 0.32
CDK6 Q00534 6/20 0.32
CCNA2 P20248 5/20 0.32
CCND1 P24385 5/20 0.32
CCND3 P30281 5/20 0.32
CCNE1 P24864 4/20 0.31
CCNH P51946 5/20 0.31
CDK1 P06493 2/20 0.31
CCNB1 P14635 2/20 0.31
MNAT1 P51948 1/20 0.31
MAPK1 P28482 1/20 0.30
HTR1A P08908 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29754894 1.00 CDK9 (0.33) CDK9CDK7CCNKCDK12CSNK1A1
SCHEMBL24676597 0.89 CDK2 (0.37) CDK9CDK7CCNKCDK12CSNK1A1
SCHEMBL29754815 0.89 CDK2 (0.37) CDK9CDK7CCNKCDK12CSNK1A1
SCHEMBL24677041 0.82 CDK6 (0.34) CDK9CDK7CCNKCDK12CSNK1A1
SCHEMBL29755036 0.81 CDK2 (0.41) CDK2CDK4CDK6CCNA2CCND1
SCHEMBL29754857 0.81 CDK2 (0.41) CDK2CDK4CDK6CCNA2CCND1
SCHEMBL24677030 0.81 CDK2 (0.41) CDK2CDK4CDK6CCNA2CCND1
SCHEMBL24675994 0.81 CDK2 (0.41) CDK2CDK4CDK6CCNA2CCND1
SCHEMBL24676684 0.80 CDK2 (0.43) CDK9CDK7CDK2CCNT1CDK4
SCHEMBL24676764 0.79 CDK2 (0.36) CDK9CDK7CCNKCDK12CSNK1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed