SCHEMBL24676714

SCHEMBL24676714

CC(C)(C)OC(=O)N1CC(c2nc(C(F)(F)F)c(-c3nc(Cl)ncc3F)s2)C1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DYRK2 Q92630 3/20 0.35
USP30 Q70CQ3 2/20 0.34
CCND1 P24385 2/20 0.34
CDK6 Q00534 2/20 0.34
NR1H2 P55055 2/20 0.33
P2RX7 Q99572 2/20 0.33
NR1H3 Q13133 1/20 0.33
MAP3K14 Q99558 1/20 0.33
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
CDK4 P11802 1/20 0.33
CCND3 P30281 1/20 0.33
TRPV3 Q8NET8 2/20 0.33
KLKB1 P03952 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
GPR119 Q8TDV5 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24676713 0.90 MAP3K14 (0.35) DYRK2USP30CCND1CDK6MAP3K14
SCHEMBL24677048 0.79 CDK2 (0.48) DYRK2CCND1CDK6CDK4CCND3
SCHEMBL29754885 0.77
SCHEMBL24676970 0.77
SCHEMBL24676727 0.76 KMT2A (0.30)
SCHEMBL29754958 0.76 ATF1 (0.31)
SCHEMBL24676744 0.76 ATF1 (0.31)
SCHEMBL24676959 0.75 DDB1 (0.37) USP30NR1H2MAP3K14TRPV3HDAC6
SCHEMBL24676513 0.75
SCHEMBL29754816 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed