SCHEMBL24676713

SCHEMBL24676713

Cc1nc(C2CN(C(=O)OC(C)(C)C)C2)sc1-c1nc(Cl)ncc1F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K14 Q99558 1/20 0.35
USP30 Q70CQ3 3/20 0.35
CCND1 P24385 3/20 0.34
CDK6 Q00534 3/20 0.34
CDK4 P11802 2/20 0.34
CCND3 P30281 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP3A5 P20815 2/20 0.34
DYRK2 Q92630 2/20 0.34
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34
PIK3CA P42336 2/20 0.33
CCNT1 O60563 1/20 0.33
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
CDK9 P50750 1/20 0.33
TRPV3 Q8NET8 2/20 0.33
KLKB1 P03952 1/20 0.33
GPR119 Q8TDV5 1/20 0.33
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24676714 0.90 DYRK2 (0.35) MAP3K14USP30CCND1CDK6CDK4
SCHEMBL24676850 0.79 CDK2 (0.49) CCND1CDK6CDK4CCND3DYRK2
SCHEMBL30926175 0.75 GPR119 (0.41) TRPV3GPR119
SCHEMBL24676013 0.75 PAX8 (0.33) USP30
SCHEMBL24675999 0.74 CDK1 (0.33) CCND1CDK6CDK4CCND3CCNT1
SCHEMBL24676849 0.72 NR1H2 (0.39) USP30PIK3CA
SCHEMBL17196760 0.72 PIK3CD (0.38) USP30CYP3A4CYP3A5GPR119
SCHEMBL17196879 0.72 PIK3CD (0.44) GPR119
SCHEMBL29611764 0.72 GRM1 (0.53) CDK9GPR119
SCHEMBL25297123 0.71 POLB (0.43) GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed