SCHEMBL24676951

SCHEMBL24676951

CNc1nc(C)c(-c2cc(NC3CCN(S(C)(=O)=O)CC3)ncc2C(F)(F)F)s1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 17/20 0.47
CCNE1 P24864 13/20 0.47
CCND1 P24385 11/20 0.43
CDK6 Q00534 11/20 0.43
CDK4 P11802 9/20 0.42
CCND3 P30281 9/20 0.42
CCNA2 P20248 4/20 0.42
CDK1 P06493 9/20 0.42
CCNB1 P14635 9/20 0.42
CCNT1 O60563 4/20 0.42
CDK9 P50750 4/20 0.42
CDK7 P50613 2/20 0.42
CCNH P51946 2/20 0.42
TDO2 P48775 1/20 0.40
IDO1 P14902 1/20 0.39
MNAT1 P51948 1/20 0.39
GPR119 Q8TDV5 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24676947 0.88 CDK2 (0.49) CDK2CCNE1CCND1CDK6CDK4
SCHEMBL24676953 0.86 CDK2 (0.47) CDK2CCNE1CCND1CDK6CDK4
SCHEMBL24676949 0.85 CDK2 (0.42) CDK2CCNE1CCND1CDK6CDK4
SCHEMBL24676827 0.84 CDK2 (0.42) CDK2CCNE1CCND1CDK6CDK4
SCHEMBL24676825 0.84 CCNA2 (0.43) CDK2CCND1CDK6CDK4CCND3
SCHEMBL24676950 0.82 TDO2 (0.42) CDK2CCNE1CCND1CDK6CDK4
SCHEMBL24676461 0.80 CDK2 (0.59) CDK2CCNE1CCND1CDK6CDK4
SCHEMBL24676948 0.79 CDK2 (0.47) CDK2CCNE1CCND1CDK6CDK4
SCHEMBL24676010 0.79 CCR6 (0.40) CDK2CCNE1CCND1CDK6CDK4
SCHEMBL29754970 0.79 CCR6 (0.40) CDK2CCNE1CCND1CDK6CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed