SCHEMBL24678728

SCHEMBL24678728

Fc1ccc(C#Cc2cnc3[nH]ccc3c2Cl)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AXL P30530 2/20 0.46
PRKCI P41743 2/20 0.46
GRM5 P41594 2/20 0.37
AAK1 Q2M2I8 2/20 0.37
ROR1 Q01973 1/20 0.34
CSNK1D P48730 1/20 0.33
MAPK14 Q16539 1/20 0.33
NUDT1 P36639 1/20 0.33
MKNK1 Q9BUB5 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33
TTBK1 Q5TCY1 3/20 0.33
TTBK2 Q6IQ55 3/20 0.33
TRPA1 O75762 2/20 0.32
MAP3K20 Q9NYL2 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
APP P05067 1/20 0.30
AURKA O14965 1/20 0.30
DAPK3 O43293 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30084172 1.00 AXL (0.46) AXLPRKCIGRM5AAK1ROR1
SCHEMBL30084219 0.86 AXL (0.48) AXLPRKCIAAK1CSNK1DMAPK14
SCHEMBL24678675 0.86 AXL (0.48) AXLPRKCIAAK1CSNK1DMAPK14
SCHEMBL24678879 0.83 AXL (0.47) AXLPRKCIAAK1CSNK1DMAPK14
SCHEMBL30084217 0.83 AXL (0.47) AXLPRKCIAAK1CSNK1DMAPK14
SCHEMBL24678177 0.82 AXL (0.49) AXLPRKCIGRM5AAK1NUDT1
SCHEMBL30084244 0.82 AXL (0.49) AXLPRKCIGRM5AAK1NUDT1
SCHEMBL24678393 0.81 AXL (0.55) AXLPRKCIGRM5AAK1CSNK1D
SCHEMBL24678122 0.81 AXL (0.48) AXLPRKCIAAK1CSNK1DMAPK14
SCHEMBL24678406 0.81 AXL (0.48) AXLPRKCIAAK1NUDT1TTBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022247676-A1 COMPOUND WITH DIPYRROLOPYRIDINE STRUCTURE, AND PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 南京康屹生物医药中心(有限合伙) 2022-12-01 WO disclosed
CN-115385911-A Compound with dipyrrolopyridine structure, preparation method and medical application 南京康屹生物医药中心(有限合伙) 2022-11-25 CN disclosed
CN-113292561-A Compound with dipyrrolopyridine structure, preparation method and medical application 中国药科大学 2021-08-24 CN disclosed