SCHEMBL24685352

SCHEMBL24685352

Cc1ccc(C2(C)CCNC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 4/20 0.53
SLC6A3 Q01959 4/20 0.53
SLC6A4 P31645 3/20 0.53
CYP2D6 P10635 1/20 0.53
OPRM1 P35372 2/20 0.45
KCNH2 Q12809 1/20 0.41
HTR2A P28223 1/20 0.38
GABRD O14764 1/20 0.38
GABRA1 P14867 1/20 0.38
GABRB1 P18505 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38
GABRA2 P47869 1/20 0.38
GABRB2 P47870 1/20 0.38
GABRA4 P48169 1/20 0.38
CHRNA1 P02708 1/20 0.38
CHRNG P07510 1/20 0.38
CHRNB1 P11230 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14390151 1.00 SLC6A2 (0.53) SLC6A2SLC6A3SLC6A4CYP2D6OPRM1
SCHEMBL18296314 0.88 OPRM1 (0.51) SLC6A2SLC6A3SLC6A4CYP2D6OPRM1
Hydrochloric Acid SCHEMBL26117908 0.86 OPRM1 (0.50) SLC6A2SLC6A3SLC6A4CYP2D6OPRM1
SCHEMBL13959656 0.82 DRD2 (0.52) SLC6A2SLC6A3SLC6A4CYP2D6HTR2A
SCHEMBL19074637 0.82 SLC6A2 (0.51) SLC6A2SLC6A3SLC6A4CYP2D6OPRM1
SCHEMBL27225389 0.82 HTR2A (0.59) SLC6A2SLC6A3SLC6A4CYP2D6OPRM1
SCHEMBL4331091 0.82 HTR2A (0.59) SLC6A2SLC6A3SLC6A4CYP2D6OPRM1
SCHEMBL27099782 0.82 HTR2A (0.59) SLC6A2SLC6A3SLC6A4CYP2D6OPRM1
Hydrochloric Acid SCHEMBL5874274 0.77 CYP2D6 (0.46) SLC6A2SLC6A3SLC6A4CYP2D6HTR2A
Hydrochloric Acid SCHEMBL5874148 0.77 CYP2D6 (0.46) SLC6A2SLC6A3SLC6A4CYP2D6HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024107393-A1 TRICYCLIC COMPOUNDS SCHRÖDINGER, INC. (US) 2024-05-23 WO disclosed
WO-2022167867-A1 SUBSTITUTED CYCLIC MODULATORS OF PROTEIN PHOSPHATASE 2A (PP2A) AND METHODS USING SAME RAPPTA THERAPEUTICS OY (FI) 2022-08-11 WO disclosed