SCHEMBL24697994

SCHEMBL24697994

CNCCNC(=O)c1cccc(-c2nc(N3CCC3)nc3c2CCC3)c1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.45
SMYD2 Q9NRG4 1/20 0.41
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
WDR5 P61964 3/20 0.39
GBA1 P04062 2/20 0.38
RAD52 P43351 2/20 0.38
MAPT P10636 1/20 0.38
PARP1 P09874 2/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
GAA P10253 1/20 0.37
GFER P55789 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
GALK1 P51570 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24698899 0.91 PRKD1 (0.42) PIK3CASMYD2NPC1RAB9AMEN1
SCHEMBL24697633 0.90 PIK3CA (0.41) PIK3CASMYD2NPC1RAB9AWDR5
SCHEMBL24697549 0.89 PIK3CA (0.54) PIK3CAGBA1MEN1KMT2A
SCHEMBL24699348 0.87 SUCNR1 (0.41) PIK3CASMYD2NPC1RAB9AGBA1
SCHEMBL30016523 0.87 MTOR (0.42) PIK3CASMYD2NPC1RAB9AWDR5
SCHEMBL24698823 0.83 USP30 (0.44) PIK3CANPC1RAB9AMAPTKMT2A
SCHEMBL19623865 0.83 PIK3CA (0.50) PIK3CAMAPTMEN1KMT2A
SCHEMBL19623703 0.83 PIK3CA (0.49) PIK3CASMYD2PARP1MEN1KMT2A
SCHEMBL24698499 0.82 NPC1 (0.44) PIK3CANPC1RAB9AMAPTMEN1
SCHEMBL19623572 0.82 PIK3CA (0.49) PIK3CAPARP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed