SCHEMBL19623865

SCHEMBL19623865

CC(C)(C)CCNC(=O)c1cccc(-c2nc(N3CCOCC3)nc3c2CCC3)c1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 6/20 0.50
PDGFRB P09619 1/20 0.44
KDR P35968 1/20 0.44
MEN1 O00255 1/20 0.41
THRB P10828 1/20 0.41
KMT2A Q03164 1/20 0.41
ATM Q13315 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
PIK3CG P48736 2/20 0.40
PIK3CD O00329 1/20 0.40
RAF1 P04049 5/20 0.40
BRAF P15056 5/20 0.40
MAPT P10636 1/20 0.40
JAK2 O60674 1/20 0.39
ACHE P22303 1/20 0.39
MTOR P42345 2/20 0.39
MAP4K4 O95819 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19623703 0.88 PIK3CA (0.49) PIK3CAMEN1THRBKMT2AATM
SCHEMBL19623572 0.87 PIK3CA (0.49) PIK3CAMEN1THRBKMT2AATM
SCHEMBL19623601 0.85 PIK3CA (0.49) PIK3CAMEN1KMT2AKDM4EPIK3CG
SCHEMBL19623874 0.83 MEN1 (0.48) PIK3CAPDGFRBKDRMEN1KMT2A
SCHEMBL24697994 0.83 PIK3CA (0.45) PIK3CAMEN1KMT2AMAPT
SCHEMBL24699348 0.82 SUCNR1 (0.41) PIK3CAACHE
SCHEMBL24698899 0.82 PRKD1 (0.42) PIK3CAMEN1KMT2AMTORMAP4K4
SCHEMBL24697633 0.81 PIK3CA (0.41) PIK3CAMEN1KMT2AKDM4EALDH1A1
SCHEMBL2375701 0.80 PIK3CA (0.65) PIK3CA
SCHEMBL19623871 0.80 PIK3CA (0.47) PIK3CAKDRKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP disclosed