SCHEMBL24698494

SCHEMBL24698494

Cn1ccc2cc(-c3nc(N4CCC4)nc4c3CCC4)ccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 6/20 0.45
TGFBR1 P36897 2/20 0.42
MAP3K20 Q9NYL2 1/20 0.42
HSD11B1 P28845 1/20 0.38
PDE10A Q9Y233 1/20 0.38
ABL1 P00519 4/20 0.37
SRC P12931 4/20 0.37
PIK3CD O00329 2/20 0.37
EGFR P00533 2/20 0.37
HCK P08631 2/20 0.37
KDR P35968 2/20 0.37
PIK3CA P42336 2/20 0.37
PIK3CB P42338 2/20 0.37
MTOR P42345 2/20 0.37
PIK3CG P48736 2/20 0.37
EPHB4 P54760 2/20 0.37
PRKDC P78527 2/20 0.37
IGF1R P08069 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24698490 0.84 ABL1 (0.39) FAAHTGFBR1MAP3K20HSD11B1PDE10A
SCHEMBL29134817 0.84 ABL1 (0.39) FAAHTGFBR1MAP3K20HSD11B1PDE10A
SCHEMBL30015747 0.84 ABL1 (0.39) FAAHTGFBR1MAP3K20HSD11B1PDE10A
SCHEMBL24699087 0.80 DYRK1A (0.43) TGFBR1MAP3K20IGF1RKDM4EALDH1A1
SCHEMBL24699477 0.77 ALDH1A1 (0.47) IGF1RKDM4EALDH1A1
SCHEMBL24699409 0.77 KDM4E (0.40) IGF1RKDM4EALDH1A1
SCHEMBL24697561 0.75 CSNK1D (0.39) ABL1SRCPIK3CDEGFRHCK
SCHEMBL24698438 0.75 ROCK2 (0.45) PDE10AKDRPIK3CAIGF1R
SCHEMBL24697795 0.75 ALDH1A1 (0.40) PIK3CAIGF1RKDM4EALDH1A1
SCHEMBL24698171 0.74 ALDH1A1 (0.54) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed