SCHEMBL24698952

SCHEMBL24698952

COC1CN(c2nc3c(c(-c4ccc(C(N)=O)cc4)n2)CCC3)C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH2 P25021 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
KARS1 Q15046 1/20 0.37
GBA1 P04062 2/20 0.36
SPR P35270 1/20 0.36
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
BTK Q06187 1/20 0.35
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP1A2 P05177 1/20 0.35
GAA P10253 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
PDE10A Q9Y233 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24698868 0.87 PDE2A (0.38) HRH2HRH3KARS1GBA1PDE4D
SCHEMBL24698191 0.86 HCRTR1 (0.36) HRH2HRH3KARS1GBA1ALDH1A1
SCHEMBL24698467 0.85 IGF1R (0.37) HRH2HRH3KARS1GBA1ALDH1A1
SCHEMBL24698950 0.83 HRH3 (0.38) HRH2HRH3KARS1GBA1SPR
SCHEMBL24698078 0.83 GBA1 (0.47) HRH2HRH3GBA1ALDH1A1KDM4E
SCHEMBL24698066 0.83 GBA1 (0.44) HRH2HRH3GBA1ALDH1A1KDM4E
SCHEMBL24698533 0.82 GBA1 (0.46) GBA1ALDH1A1KDM4EGAAHPGD
SCHEMBL24698716 0.81 HRH3 (0.36) HRH2HRH3GBA1PDE4DALDH1A1
SCHEMBL24698712 0.81 HRH3 (0.36) HRH2HRH3GBA1PDE4DALDH1A1
SCHEMBL24698917 0.80 PDE10A (0.39) PDE4DALDH1A1PDE10AEEF2KPDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed