SCHEMBL24698917

SCHEMBL24698917

NC(=O)c1ccc(-c2nc(N3CC(O)C3)nc3c2CC3)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.39
PDE2A O00408 1/20 0.39
CHEK1 O14757 2/20 0.36
KDM1A O60341 1/20 0.35
IKBKB O14920 1/20 0.34
PIK3CA P42336 2/20 0.33
LCK P06239 1/20 0.33
JAK3 P52333 1/20 0.33
TBK1 Q9UHD2 1/20 0.33
PDE4D Q08499 1/20 0.33
PDE7A Q13946 1/20 0.33
PTK2 Q05397 1/20 0.32
CHUK O15111 1/20 0.32
P2RY12 Q9H244 1/20 0.32
SMO Q99835 1/20 0.32
MKNK1 Q9BUB5 2/20 0.31
MKNK2 Q9HBH9 2/20 0.31
EEF2K O00418 1/20 0.31
MAPK1 P28482 1/20 0.31
MAP2K4 P45985 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24698868 0.93 PDE2A (0.38) PDE10APDE2ACHEK1KDM1APIK3CA
SCHEMBL24699410 0.85 ALDH1A1 (0.38) CHEK1KDM1AIKBKBPIK3CAMAPK1
SCHEMBL24698191 0.82 HCRTR1 (0.36) PDE10APDE2ACHEK1KDM1APIK3CA
SCHEMBL30016847 0.82 SMO (0.36) PDE10APDE2ACHEK1KDM1APTK2
SCHEMBL24698914 0.82 SMO (0.36) PDE10APDE2ACHEK1KDM1APTK2
SCHEMBL24698426 0.82 KARS1 (0.40) PIK3CAP2RY12EEF2KALDH1A1
SCHEMBL24698467 0.81 IGF1R (0.37) PDE10APDE2AKDM1AEEF2KALDH1A1
SCHEMBL24698430 0.80 PIK3CA (0.46) PDE10AKDM1APIK3CAMAPK1MAP2K4
SCHEMBL24698078 0.79 GBA1 (0.47) CHEK1PIK3CAALDH1A1
SCHEMBL24698066 0.79 GBA1 (0.44) CHEK1KDM1APIK3CAEEF2KALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed