SCHEMBL24699239

SCHEMBL24699239

CCS(=N)(=O)c1cc(-c2nc(N3CC[C@@H]3C)nc3c2CCC3)ccc1OC

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMOX1 P09601 1/20 0.34
CA4 P22748 1/20 0.34
POLB P06746 2/20 0.34
ALDH1A1 P00352 1/20 0.34
EHMT2 Q96KQ7 4/20 0.34
LMNA P02545 1/20 0.34
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
BRD4 O60885 3/20 0.33
BRD3 Q15059 3/20 0.33
CRHR1 P34998 1/20 0.33
BRD2 P25440 1/20 0.33
HRH2 P25021 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24697981 0.92 PIK3R1 (0.36) HMOX1CA4POLBEHMT2LMNA
SCHEMBL24699240 0.89 MTOR (0.35) MTOR
SCHEMBL30015790 0.87 MTOR (0.32) POLBEHMT2LMNACA12CA2
SCHEMBL24698640 0.87 MTOR (0.32) POLBEHMT2LMNACA12CA2
SCHEMBL24699603 0.86 BRD4 (0.37) CA4POLBEHMT2CA12CA1
SCHEMBL30016531 0.84 PI4KB (0.36) ALDH1A1CA12CA1CA2CA9
SCHEMBL24697976 0.84 PI4KB (0.36) ALDH1A1CA12CA1CA2CA9
SCHEMBL24699229 0.84 MTOR (0.36) LMNAPDK1PDK2PDK3PDK4
SCHEMBL30016058 0.84 MTOR (0.36) LMNAPDK1PDK2PDK3PDK4
SCHEMBL24699069 0.83 PI4KB (0.35) POLBPDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed