SCHEMBL24699345

SCHEMBL24699345

C[C@H]1CCN1c1nc2c(c(-c3cccc(C(=O)NCCNC(=O)OC(C)(C)C)c3)n1)CCC2

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACACB O00763 2/20 0.41
ACACA Q13085 2/20 0.41
MTOR P42345 4/20 0.40
USP30 Q70CQ3 1/20 0.39
SUCNR1 Q9BXA5 2/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
NAMPT P43490 2/20 0.37
GABRA5 P31644 1/20 0.37
SYK P43405 2/20 0.36
CKS1B P61024 1/20 0.36
SKP1 P63208 1/20 0.36
SKP2 Q13309 1/20 0.36
MLLT1 Q03111 1/20 0.36
PIK3R1 P27986 1/20 0.35
PIK3CA P42336 1/20 0.35
SMYD2 Q9NRG4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30016077 1.00 ACACB (0.41) ACACBACACAMTORUSP30SUCNR1
SCHEMBL24699348 0.88 SUCNR1 (0.41) ACACBACACAUSP30SUCNR1NPC1
SCHEMBL30016523 0.88 MTOR (0.42) MTORNPC1RAB9ASYKPIK3R1
SCHEMBL24698892 0.88 MTOR (0.48) MTORNPC1RAB9ASYKSMYD2
SCHEMBL24697628 0.88 MTOR (0.42) MTORNPC1RAB9ASYKPIK3CA
SCHEMBL30016136 0.87 ROCK2 (0.43) ACACBACACAMTORNAMPTCKS1B
SCHEMBL29134944 0.87 ROCK2 (0.43) ACACBACACAMTORNAMPTCKS1B
SCHEMBL24698512 0.87 ROCK2 (0.43) ACACBACACAMTORNAMPTCKS1B
SCHEMBL24697681 0.87 HRH3 (0.42) MTORNPC1RAB9ASYKSMYD2
SCHEMBL30017041 0.87 HRH3 (0.42) MTORNPC1RAB9ASYKSMYD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed