SCHEMBL24699359

SCHEMBL24699359

CN1C(=O)N[C@]2(CCc3cc(Br)ccc32)C1=O

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 10/20 0.48
BRD4 O60885 1/20 0.41
AKR1B1 P15121 1/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
POLB P06746 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30016504 1.00 BACE1 (0.48) BACE1BRD4AKR1B1LMNAHPGD
SCHEMBL449103 0.82 AKR1B1 (0.50) BACE1AKR1B1LMNAHPGDHTT
SCHEMBL30297507 0.80 TSHR (0.56) AKR1B1LMNAHPGDPOLBHSD17B10
SCHEMBL445231 0.80 BACE1 (0.49) BACE1AKR1B1
SCHEMBL1814392 0.78 BACE1 (0.51) BACE1BRD4LMNAHTTMAPT
SCHEMBL17605103 0.77 KMT2A (0.53) LMNAPOLBMEN1MAPTKMT2A
SCHEMBL21132278 0.76 LMNA (0.41) LMNAHPGDPOLBHSD17B10MEN1
SCHEMBL1978797 0.76 BACE1 (0.46) BACE1AKR1B1MAPT
SCHEMBL17606047 0.75 TSHR (0.63) AKR1B1
SCHEMBL17606065 0.75 TSHR (0.63) AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed