SCHEMBL24699403

SCHEMBL24699403

C[C@H]1[C@H](O)CN1c1nc2c(c(-c3ccc(-c4ncc[nH]4)cc3)n1)CCC2

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.36
MTOR P42345 5/20 0.35
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
ADK P55263 1/20 0.32
HRH3 Q9Y5N1 2/20 0.32
KCNH2 Q12809 1/20 0.32
HRH2 P25021 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP19A1 P11511 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24699404 0.84 NISCH (0.35) NISCHMTORKDM4EALDH1A1ADK
SCHEMBL24698946 0.83 MTOR (0.42) NISCHMTORKDM4EALDH1A1ADK
SCHEMBL24698948 0.79 NISCH (0.38) NISCHMTORKDM4EALDH1A1ADK
SCHEMBL24698425 0.79 MEN1 (0.37) KDM4EHRH3HRH2
SCHEMBL24698179 0.79 WNT3A (0.36) HRH3HRH2
SCHEMBL24699434 0.79 HRH2 (0.39) ALDH1A1HRH3HRH2
SCHEMBL24697597 0.78 HRH2 (0.36) MTORKDM4EALDH1A1HRH3HRH2
SCHEMBL24698865 0.78 HRH2 (0.36) MTORKDM4EALDH1A1HRH3HRH2
SCHEMBL24698116 0.77 HRH3 (0.35) ALDH1A1HRH3KCNH2HRH2
SCHEMBL24699039 0.77 KHK (0.36) HRH3HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4313967-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-07 EP disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed