SCHEMBL24699404

SCHEMBL24699404

OC1CN(c2nc3c(c(-c4ccc(-c5ncc[nH]5)cc4)n2)CCC3)C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.35
KDM4E B2RXH2 6/20 0.35
ALDH1A1 P00352 3/20 0.35
MAPT P10636 2/20 0.35
TP53 P04637 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MTOR P42345 5/20 0.34
ADK P55263 1/20 0.34
HRH3 Q9Y5N1 2/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
KCNH2 Q12809 1/20 0.33
TBK1 Q9UHD2 1/20 0.33
LMNA P02545 2/20 0.32
USP2 O75604 1/20 0.32
HPGD P15428 1/20 0.32
MAPK1 P28482 1/20 0.32
HSD17B10 Q99714 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HRH2 P25021 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24698948 0.86 NISCH (0.38) NISCHKDM4EALDH1A1L3MBTL1MTOR
SCHEMBL24699403 0.84 NISCH (0.36) NISCHKDM4EALDH1A1MTORADK
SCHEMBL24698946 0.80 MTOR (0.42) NISCHKDM4EALDH1A1MTORADK
SCHEMBL24698426 0.77 KARS1 (0.40) KDM4EALDH1A1MTORHRH3HCRTR1
SCHEMBL24698113 0.77 HRH2 (0.36) KDM4EALDH1A1MAPTTP53L3MBTL1
SCHEMBL24699432 0.77 HRH2 (0.38) KDM4EALDH1A1MAPTTP53L3MBTL1
SCHEMBL24698868 0.76 PDE2A (0.38) KDM4EALDH1A1HRH3HCRTR1HCRTR2
SCHEMBL24698181 0.76 GBA1 (0.38) KDM4EALDH1A1MAPTTP53L3MBTL1
SCHEMBL24699006 0.75 KDM4E (0.39) KDM4EALDH1A1HPGDHSD17B10
SCHEMBL24698195 0.75 PRKACA (0.38) KDM4EMAPTTP53L3MBTL1TBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed