SCHEMBL24699485

SCHEMBL24699485

COc1cc(-c2nc(N3CCC3)nc3c2CCC3)ccc1C(N)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.42
ALDH1A1 P00352 4/20 0.42
HPGD P15428 4/20 0.42
TP53 P04637 1/20 0.42
GAA P10253 1/20 0.42
MKNK1 Q9BUB5 2/20 0.42
MKNK2 Q9HBH9 2/20 0.42
TGFBR1 P36897 1/20 0.41
ACVR1 Q04771 1/20 0.41
HSD17B10 Q99714 4/20 0.40
MAPK1 P28482 2/20 0.40
TSHR P16473 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NEK2 P51955 1/20 0.40
EHMT2 Q96KQ7 1/20 0.40
EHMT1 Q9H9B1 1/20 0.40
GBA1 P04062 1/20 0.40
DHFR P00374 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24698964 0.89 MKNK1 (0.44) KDM4EALDH1A1HPGDTP53GAA
SCHEMBL24699484 0.86 PDE7A (0.41) KDM4EALDH1A1HPGDMKNK1MKNK2
SCHEMBL30015689 0.86 PDE7A (0.41) KDM4EALDH1A1HPGDMKNK1MKNK2
SCHEMBL24699356 0.85 GBA1 (0.47) KDM4EALDH1A1HPGDTP53GAA
SCHEMBL24699459 0.84 GBA1 (0.39) KDM4EALDH1A1HPGDTP53GAA
SCHEMBL24699476 0.84 GBA1 (0.39) KDM4EALDH1A1HPGDTP53GAA
SCHEMBL24698767 0.82 GBA1 (0.38) KDM4EALDH1A1HPGDTP53GAA
SCHEMBL24699054 0.81 GBA1 (0.38) KDM4EALDH1A1HPGDTP53GAA
SCHEMBL24699497 0.80 HSD17B10 (0.43) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL24698066 0.79 GBA1 (0.44) KDM4EALDH1A1HPGDTP53GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed