SCHEMBL24699484

SCHEMBL24699484

COc1cc(-c2nc(N3CC[C@@H]3C)nc3c2CCC3)ccc1C(N)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 1/20 0.41
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
PDK1 Q15118 1/20 0.39
PDK2 Q15119 1/20 0.39
PDK3 Q15120 1/20 0.39
PDK4 Q16654 1/20 0.39
EHMT2 Q96KQ7 1/20 0.39
MTOR P42345 3/20 0.38
TGFBR1 P36897 1/20 0.37
ACVR1 Q04771 1/20 0.37
PARP15 Q460N3 1/20 0.37
PARP10 Q53GL7 1/20 0.37
DHFR P00374 2/20 0.37
NEK2 P51955 1/20 0.36
GAK O14976 1/20 0.36
HSD17B10 Q99714 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30015689 1.00 PDE7A (0.41) PDE7AMKNK1MKNK2PDK1PDK2
SCHEMBL24698959 0.90 MKNK1 (0.42) MKNK1MKNK2PDK1PDK2PDK3
SCHEMBL30014971 0.90 MKNK1 (0.42) MKNK1MKNK2PDK1PDK2PDK3
SCHEMBL30015877 0.87 PDK1 (0.40) MKNK1MKNK2PDK1PDK2PDK3
SCHEMBL24699461 0.87 PDK1 (0.40) MKNK1MKNK2PDK1PDK2PDK3
SCHEMBL30016341 0.87 MTOR (0.44) PDK1PDK2PDK3PDK4MTOR
SCHEMBL24699474 0.87 MTOR (0.44) PDK1PDK2PDK3PDK4MTOR
SCHEMBL24699353 0.86 PDK1 (0.39) PDE7APDK1PDK2PDK3PDK4
SCHEMBL24699485 0.86 KDM4E (0.42) PDE7AMKNK1MKNK2EHMT2TGFBR1
SCHEMBL30015382 0.86 PDK1 (0.39) PDE7APDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed