SCHEMBL247092

SCHEMBL247092

OC[C@H](O)Cc1ccc(Cl)cc1Cl

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 6/20 0.48
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 2/20 0.42
GGPS1 O95749 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
HDAC8 Q9BY41 3/20 0.41
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
ACLY P53396 3/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL247767 1.00 IDO1 (0.48) IDO1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL10325517 1.00 IDO1 (0.48) IDO1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL3237063 0.83 IDO1 (0.47) IDO1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL10587518 0.83 IDO1 (0.47) IDO1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL3437067 0.83 IDO1 (0.47) IDO1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL250266 0.81 ACLY (0.47) IDO1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL22145306 0.81 PYCR1 (0.40) IDO1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL11471881 0.81 ACLY (0.47) IDO1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL15066555 0.81 ACLY (0.47) IDO1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8422598 0.80 IDO1 (0.52) IDO1CYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2968210-A1 PHENYL CARBAMATE COMPOUNDS FOR USE IN PREVENTING OR TREATING PEDIATRIC EPILESY AND EPILESY-RELATED SYNDROMES Bio-Pharm Solutions Co., Ltd. (KR) 2016-01-20 EP disclosed
EP-2970110-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR PREVENTING OR TREATING A PSYCHIATRIC DISORDER COMPRISING THE SAME Bio-Pharm Solutions Co., Ltd. (KR) 2016-01-20 EP disclosed
EP-2970112-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR PREVENTING OR TREATING A MEMORY LOSS-RELATED DISEASE COMPRISING THE SAME Bio-Pharm Solutions Co., Ltd. (KR) 2016-01-20 EP disclosed
WO-2014142549-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR PREVENTING OR TREATING A MEMORY LOSS-RELATED DISEASE COMPRISING THE SAME BIO-PHARM SOLUTIONS CO., LTD. (KR) 2014-09-18 WO disclosed
WO-2014142477-A1 PHENYL CARBAMATE COMPOUNDS FOR USE IN PREVENTING OR TREATING PEDIATRIC EPILESY AND EPILESY-RELATED SYNDROMES BIO-PHARM SOLUTIONS CO., LTD. (KR) 2014-09-18 WO disclosed
WO-2014142550-A1 PHENYL CARBAMATE COMPOUND AND A COMPOSITION FOR PREVENTING OR TREATING A PSYCHIATRIC DISORDER COMPRISING THE SAME BIO-PHARM SOLUTIONS CO., LTD. (KR) 2014-09-18 WO disclosed
EP-2590936-A2 PHENYLCARBAMATE COMPOUND AND MUSCLE RELAXANT CONTAINING THE SAME Bio-Pharm Solutions Co., Ltd. (KR) 2013-05-15 EP disclosed
WO-2012002773-A2 PHENYLCARBAMATE COMPOUND AND MUSCLE RELAXANT CONTAINING THE SAME BIO-PHARM SOLUTIONS CO., LTD. (KR) 2012-01-05 WO disclosed