SCHEMBL2470985

SCHEMBL2470985

C=CCN(CC=C)CCc1ccc(NS(=O)(=O)c2ccc(C(C)C)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
MAPT P10636 2/20 0.50
LMNA P02545 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
PKM P14618 1/20 0.50
GHSR Q92847 1/20 0.47
ADRB2 P07550 3/20 0.46
ADRB1 P08588 3/20 0.46
ADRB3 P13945 3/20 0.46
DRD2 P14416 1/20 0.46
DRD3 P35462 1/20 0.46
KCNH2 Q12809 1/20 0.46
PGR P06401 1/20 0.43
POLB P06746 1/20 0.43
THRB P10828 1/20 0.43
FFAR1 O14842 1/20 0.43
FFAR4 Q5NUL3 1/20 0.43
TRIM24 O15164 1/20 0.42
BRD1 O95696 1/20 0.42
BRPF1 P55201 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4920272 0.99 ALDH1A1 (0.49) ALDH1A1MAPTLMNASMN1; SMN2PKM
SCHEMBL2466084 0.84 FFAR1 (0.51) ALDH1A1MAPTLMNASMN1; SMN2PKM
Hydrochloric Acid SCHEMBL4914708 0.83 FFAR1 (0.50) ALDH1A1MAPTLMNASMN1; SMN2PKM
SCHEMBL2470496 0.82 ADRB2 (0.57) ALDH1A1MAPTLMNASMN1; SMN2PKM
SCHEMBL1719317 0.82 DRD3 (0.42) DRD2DRD3KCNH2
Hydrochloric Acid SCHEMBL4915819 0.81 ADRB2 (0.56) ALDH1A1MAPTLMNASMN1; SMN2PKM
Hydrochloric Acid SCHEMBL4918974 0.81 DRD3 (0.42) DRD2DRD3KCNH2
SCHEMBL2472476 0.81 ADRB3 (0.51) ALDH1A1MAPTLMNASMN1; SMN2PKM
SCHEMBL2473909 0.79 HDAC1 (0.49) MAPTSMN1; SMN2DRD2DRD3KCNH2
Hydrochloric Acid SCHEMBL4919634 0.78 HDAC1 (0.48) MAPTSMN1; SMN2DRD2DRD3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2371814-A1 Aminoethylaromatic compounds suitable for treating disorders that respond to modulation of the dopamine D3 receptor Abbott GmbH & Co. KG (DE) 2011-10-05 EP disclosed
EP-1809597-A1 AMINOETHYLAROMATIC COMPOUNDS SUITABLE FOR TREATING DISORDERS THAT RESPOND TO MODULATION OF THE DOPAMINE D3 RECEPTOR Abbott GmbH & Co. KG (DE) 2007-07-25 EP disclosed
WO-2006040179-A1 AMINOETHYLAROMATIC COMPOUNDS SUITABLE FOR TREATING DISORDERS THAT RESPOND TO MODULATION OF THE DOPAMINE D3 RECEPTOR ABBOTT GMBH & CO. KG (DE) 2006-04-20 WO disclosed