SCHEMBL24710459

SCHEMBL24710459

Cc1ccnn(C2=CN(C(=O)OC(C)(C)C)CCC2)c1=O

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 1/20 0.36
MCHR1 Q99705 1/20 0.36
GPR119 Q8TDV5 5/20 0.36
SPR P35270 1/20 0.35
GRM5 P41594 1/20 0.34
BTK Q06187 1/20 0.33
TP53 P04637 1/20 0.33
DTYMK P23919 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
POLB P06746 1/20 0.33
GRM1 Q13255 1/20 0.32
ELANE P08246 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24710878 0.81 GRM5 (0.33) GPR119SPRGRM5BTKTP53
SCHEMBL24710633 0.76 GPR119 (0.34) GPR119GRM5BTKDTYMKPOLB
SCHEMBL24711551 0.74 GPR119 (0.37) GPR119SPRGRM5BTKKMT2A
SCHEMBL975177 0.74 HPGD (0.37) GPR119BTKMEN1KMT2A
SCHEMBL14878683 0.72 USP2 (0.39) GPR119GRM5BTKMEN1KMT2A
SCHEMBL12538830 0.71 BTK (0.40) GPR119GRM5BTKMEN1KMT2A
SCHEMBL21258531 0.71 BTK (0.36) GPR119GRM5BTKDTYMKMEN1
SCHEMBL31555855 0.70 BTK (0.47) GPR119GRM5BTKMEN1KMT2A
SCHEMBL4762097 0.69 USP2 (0.41) GPR119GRM5BTKMEN1KMT2A
SCHEMBL7899134 0.68 USP2 (0.38) GPR119BTKMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022258986-A1 COMPOUNDS USEFUL IN THE TREATMENT OR PREVENTION OF A PRMT5-MEDIATED DISORDER Argonaut Therapeutics Limited (GB) 2022-12-15 WO disclosed