SCHEMBL2471315

SCHEMBL2471315

Oc1cccc(C#Cc2cccc3ccccc23)c1O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.54
PTPN22 Q9Y2R2 1/20 0.50
CHAT P28329 1/20 0.47
GRM5 P41594 1/20 0.44
POLB P06746 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ALDH1A1 P00352 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
HSD17B10 Q99714 2/20 0.41
ADAMTS4 O75173 1/20 0.41
EGFR P00533 1/20 0.41
LMNA P02545 1/20 0.41
FYN P06241 1/20 0.41
MMP2 P08253 1/20 0.41
MMP9 P14780 1/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41
MMP8 P22894 1/20 0.41
CA6 P23280 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2474670 0.88 CYP1A2 (0.58) CYP1A2PTPN22CHATGRM5POLB
SCHEMBL2477460 0.85 CYP1A2 (0.54) CYP1A2PTPN22CHATGRM5POLB
SCHEMBL2776015 0.83 CHAT (0.60) CYP1A2CHATGRM5POLBALDH1A1
SCHEMBL29661843 0.83 CHAT (0.60) CYP1A2CHATGRM5POLBALDH1A1
SCHEMBL6364668 0.81 CHAT (0.58) CYP1A2CHATGRM5POLBALDH1A1
SCHEMBL28797628 0.78 PTPN22 (0.47) CYP1A2PTPN22CHATGRM5POLB
SCHEMBL2473787 0.77 CHAT (0.44) CYP1A2PTPN22CHATGRM5POLB
SCHEMBL951002 0.76 ALDH1A1 (0.50) CYP1A2GRM5ALDH1A1CA1CA2
SCHEMBL2474672 0.76 CHAT (0.58) CYP1A2CHATGRM5POLBL3MBTL1
SCHEMBL5881381 0.75 CHAT (0.49) CYP1A2PTPN22CHATGRM5POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2373721-B1 ACETYLENIC AROMATIC POLYETHERKETONE NEXAM CHEMICAL AB (SE) 2014-06-25 EP disclosed
EP-2373721-A1 ACETYLENIC AROMATIC POLYETHERKETONE Nexam Chemical AB (SE) 2011-10-12 EP disclosed
WO-2010072760-A1 ACETYLENIC AROMATIC POLYETHERKETONE NEXAM CHEMICAL AB (SE) 2010-07-01 WO disclosed