SCHEMBL24714950

SCHEMBL24714950

C=CC(=O)Nc1cc2c(Nc3cc(-c4ccc(F)cc4F)ccc3OC)ncnc2cc1N1CCC(N2CCOCC2)CC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 19/20 0.55
KDR P35968 6/20 0.46
ERBB3 P21860 3/20 0.46
DUS2 Q9NX74 1/20 0.46
ERBB2 P04626 3/20 0.45
KIT P10721 2/20 0.45
SRC P12931 2/20 0.45
ERBB4 Q15303 2/20 0.45
IRAK4 Q9NWZ3 2/20 0.45
BMPR1B O00238 1/20 0.45
CIT O14578 1/20 0.45
MAP2K7 O14733 1/20 0.45
GAK O14976 1/20 0.45
EPHB6 O15197 1/20 0.45
MAP3K7 O43318 1/20 0.45
RIPK2 O43353 1/20 0.45
STK17B O94768 1/20 0.45
STK10 O94804 1/20 0.45
ABL1 P00519 1/20 0.45
LCK P06239 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30030882 1.00 EGFR (0.55) EGFRKDRERBB3DUS2ERBB2
SCHEMBL27139860 0.86 EGFR (0.53) EGFRKDRERBB3DUS2
SCHEMBL24713933 0.86 EGFR (0.51) EGFRKDRERBB3DUS2
SCHEMBL30822153 0.86 EGFR (0.49) EGFRKDRERBB3DUS2ERBB2
SCHEMBL24714506 0.86 EGFR (0.49) EGFRKDRERBB3DUS2ERBB2
SCHEMBL24714723 0.85 EGFR (0.52) EGFRKDRERBB3DUS2
SCHEMBL27136337 0.85 EGFR (0.51) EGFRKDRERBB3DUS2
SCHEMBL24714969 0.83 EGFR (0.63) EGFRKDRERBB3DUS2SRC
SCHEMBL30031056 0.79 EGFR (0.60) EGFRERBB2SRCERBB4GAK
SCHEMBL24714972 0.79 EGFR (0.60) EGFRERBB2SRCERBB4GAK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4328222-A1 HETEROARYL DERIVATIVE COMPOUND AND USE THEREOF Voronoi Inc. (KR) 2024-02-28 EP claimed
EP-4328222-A1 HETEROARYL DERIVATIVE COMPOUND AND USE THEREOF Voronoi Inc. (KR) 2024-02-28 EP disclosed
WO-2022225238-A1 HETEROARYL DERIVATIVE COMPOUND AND USE THEREOF 보로노이 주식회사 2022-10-27 WO disclosed