SCHEMBL27136337

SCHEMBL27136337

C=CC(=O)Nc1cc2c(Nc3cc(-c4ccc(F)cc4F)ccc3OC)ncnc2cc1N1CC(F)(F)C1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.51
ERBB3 P21860 1/20 0.49
DUS2 Q9NX74 1/20 0.49
KDR P35968 16/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27139860 0.93 EGFR (0.53) EGFRERBB3DUS2KDR
SCHEMBL24714506 0.92 EGFR (0.49) EGFRERBB3DUS2KDR
SCHEMBL30822153 0.92 EGFR (0.49) EGFRERBB3DUS2KDR
SCHEMBL24714723 0.90 EGFR (0.52) EGFRERBB3DUS2KDR
SCHEMBL24713933 0.90 EGFR (0.51) EGFRERBB3DUS2KDR
SCHEMBL24714969 0.87 EGFR (0.63) EGFRERBB3DUS2KDR
SCHEMBL30030882 0.85 EGFR (0.55) EGFRERBB3DUS2KDR
SCHEMBL24714950 0.85 EGFR (0.55) EGFRERBB3DUS2KDR
SCHEMBL24714738 0.83 EGFR (0.49) EGFRKDR
SCHEMBL24715219 0.80 EGFR (0.50) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4328222-A1 HETEROARYL DERIVATIVE COMPOUND AND USE THEREOF Voronoi Inc. (KR) 2024-02-28 EP claimed
US-20240246940-A1 HETEROARYL DERIVATIVE COMPOUND AND USE THEREOF VORONOI INC. (KR) 2024-07-25 US disclosed
EP-4328222-A1 HETEROARYL DERIVATIVE COMPOUND AND USE THEREOF Voronoi Inc. (KR) 2024-02-28 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240246940-A1 HETEROARYL DERIVATIVE COMPOUND AND USE THEREOF ERBB2, EGFR, ERBB3 EGFR 2/4885ERBB3 3/4885DUS2 2381/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.