SCHEMBL24717540

SCHEMBL24717540

CO[C@H]1C[C@H](N2CCC[C@@H](O)C2)C1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.34
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
CCR4 P51679 1/20 0.33
ADRA1A P35348 1/20 0.33
ALDH1A1 P00352 1/20 0.33
DPP4 P27487 1/20 0.32
DPP8 Q6V1X1 1/20 0.32
DPP9 Q86TI2 1/20 0.32
MAN2B1 O00754 1/20 0.32
KDM2B Q8NHM5 1/20 0.31
GRM3 Q14832 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24717539 1.00 HRH3 (0.34) HRH3CA12CA1CA2CA9
SCHEMBL24717795 0.83 HRH3 (0.42) HRH3CCR4ADRA1AALDH1A1DPP4
SCHEMBL24717794 0.83 HRH3 (0.42) HRH3CCR4ADRA1AALDH1A1DPP4
SCHEMBL26936208 0.80 ADRA1A (0.40) HRH3ADRA1AALDH1A1
SCHEMBL29335361 0.79 HRH3 (0.34) HRH3
SCHEMBL24718209 0.79 HRH3 (0.34) HRH3
SCHEMBL24718208 0.77 GAA (0.32)
SCHEMBL24718203 0.77 GAA (0.32)
SCHEMBL2618405 0.77 HRH3 (0.37) HRH3CCR4ADRA1AALDH1A1KDM2B
SCHEMBL29335376 0.77 LMNA (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220395576-A1 MODULATORS OF BCL6 PROTEOLYSIS AND ASSOCIATED METHODS OF USE ARVINAS OPERATIONS, INC. 2022-12-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220395576-A1 MODULATORS OF BCL6 PROTEOLYSIS AND ASSOCIATED METHODS OF USE BCL6, BCL6B, BCL3 HRH3 3492/4885CA12 3307/4885CA1 2454/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.