SCHEMBL24720649

SCHEMBL24720649

Cc1cc(-c2ccc(C)c(C)c2)c(O)c(-c2ccc(N)c(Cl)c2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.47
CYP3A4 P08684 7/20 0.46
ALDH1A1 P00352 5/20 0.46
TSHR P16473 4/20 0.46
MAPK1 P28482 1/20 0.46
TDP1 Q9NUW8 1/20 0.39
MAPT P10636 2/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
AKR1C2 P52895 1/20 0.34
AKR1C1 Q04828 1/20 0.34
PTGS1 P23219 2/20 0.33
PTGS2 P35354 2/20 0.33
MCL1 Q07820 1/20 0.33
THRB P10828 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
CASP1 P29466 1/20 0.33
RECQL P46063 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24720587 0.91 ESR2 (0.47) ESR2CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL24720257 0.84 ESR2 (0.41) ESR2CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL24720574 0.83 ESR2 (0.40) ESR2CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL24720935 0.80 ESR2 (0.43) ESR2CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL24719632 0.80 ESR2 (0.43) ESR2CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL24721426 0.77 TNKS2 (0.40) ESR2CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL26976338 0.73 CYP3A4 (0.74) ESR2CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL26976337 0.71 CYP3A4 (0.71) ESR2CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL22453110 0.70 TSHR (0.55) ESR2CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL24720517 0.69 TLR8 (0.45) ESR2ALDH1A1MAPTPTGS2MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022261204-A1 ANTICANCER COMPOUNDS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-12-15 WO disclosed