SCHEMBL24720587

SCHEMBL24720587

Cc1cc(-c2ccc(Cl)c(C)c2)c(O)c(-c2ccc(N)c(Cl)c2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.47
CYP3A4 P08684 5/20 0.46
ALDH1A1 P00352 4/20 0.46
TSHR P16473 4/20 0.46
MAPK1 P28482 1/20 0.46
TDP1 Q9NUW8 1/20 0.39
PTGS2 P35354 3/20 0.39
PTGS1 P23219 2/20 0.39
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
CD44 P16070 1/20 0.35
AKR1C2 P52895 2/20 0.34
AKR1C1 Q04828 1/20 0.34
AKR1C3 P42330 1/20 0.34
SRC P12931 1/20 0.33
ALKBH3 Q96Q83 1/20 0.33
AHR P35869 1/20 0.33
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24720649 0.91 ESR2 (0.47) ESR2CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL24720257 0.84 ESR2 (0.41) ESR2CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL24720574 0.83 ESR2 (0.40) ESR2CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL24719632 0.80 ESR2 (0.43) ESR2CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL24720935 0.80 ESR2 (0.43) ESR2CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL24721426 0.77 TNKS2 (0.40) ESR2CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL24720518 0.74 LRRK2 (0.40) ESR2CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL5845416 0.74 CYP3A4 (0.63) ESR2CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL26976338 0.73 CYP3A4 (0.74) ESR2CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL26327407 0.72 PTGS2 (0.43) PTGS2PTGS1AKR1C2AKR1C3ALKBH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022261204-A1 ANTICANCER COMPOUNDS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-12-15 WO disclosed