SCHEMBL24720935

SCHEMBL24720935

Cc1cncc(-c2cc(C)cc(-c3ccc(N)c(Cl)c3)c2O)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.43
ALDH1A1 P00352 2/20 0.41
CYP3A4 P08684 2/20 0.41
TSHR P16473 2/20 0.41
MAPK1 P28482 1/20 0.41
PTGS2 P35354 1/20 0.38
CYP2A6 P11509 3/20 0.37
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
TDO2 P48775 1/20 0.33
ACLY P53396 2/20 0.33
GSK3B P49841 1/20 0.33
PIK3CD O00329 1/20 0.33
GYS1 P13807 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24720257 0.82 ESR2 (0.41) ESR2ALDH1A1CYP3A4TSHRMAPK1
SCHEMBL24720649 0.80 ESR2 (0.47) ESR2ALDH1A1CYP3A4TSHRMAPK1
SCHEMBL24720587 0.80 ESR2 (0.47) ESR2ALDH1A1CYP3A4TSHRMAPK1
SCHEMBL24719632 0.78 ESR2 (0.43) ESR2ALDH1A1CYP3A4TSHRMAPK1
SCHEMBL24720518 0.78 LRRK2 (0.40) ESR2ALDH1A1CYP3A4TSHRMAPK1
SCHEMBL24721413 0.74 PTGS2 (0.33) PTGS2ACLY
SCHEMBL24721426 0.73 TNKS2 (0.40) ESR2ALDH1A1CYP3A4TSHRMAPK1
SCHEMBL24720574 0.73 ESR2 (0.40) ESR2ALDH1A1CYP3A4TSHRMAPK1
SCHEMBL24721356 0.69 ESR2 (0.45) ESR2ALDH1A1CYP3A4TSHRMAPK1
SCHEMBL7088612 0.68 CYP2A6 (0.46) ALDH1A1CYP3A4TSHRPTGS2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022261204-A1 ANTICANCER COMPOUNDS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-12-15 WO disclosed