SCHEMBL2472263

SCHEMBL2472263

CCc1ccc(CCNC(=O)C2(Cc3ccccc3)CCN(S(=O)(=O)c3ccc(C)cc3)CC2)cc1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.59
KMT2A Q03164 5/20 0.59
GAA P10253 4/20 0.57
POLB P06746 1/20 0.57
MAPT P10636 1/20 0.57
HTT P42858 1/20 0.57
ALDH1A1 P00352 3/20 0.54
FKBP1A P62942 1/20 0.52
HSD11B1 P28845 1/20 0.49
CYP2C19 P33261 1/20 0.48
PKM P14618 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2472232 0.94 GAA (0.54) MEN1KMT2AGAAPOLBMAPT
SCHEMBL2469016 0.91 KMT2A (0.51) MEN1KMT2AGAAPOLBMAPT
SCHEMBL2472160 0.91 FKBP1A (0.51) MEN1KMT2AGAAPOLBMAPT
SCHEMBL2469084 0.90 KMT2A (0.61) MEN1KMT2AGAAPOLBMAPT
SCHEMBL2465751 0.87 MEN1 (0.50) MEN1KMT2AGAAPOLBMAPT
SCHEMBL2471923 0.87 TP53 (0.47) MEN1KMT2APOLBALDH1A1FKBP1A
SCHEMBL2465689 0.86 ALDH1A1 (0.52) MEN1KMT2AGAAPOLBMAPT
SCHEMBL2471780 0.83 MEN1 (0.55) MEN1KMT2AGAAALDH1A1FKBP1A
SCHEMBL2470282 0.82 ALDH1A1 (0.48) MEN1KMT2APOLBMAPTHTT
SCHEMBL2473023 0.82 FKBP1A (0.44) MEN1KMT2AGAAMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2371366-A1 Heterocyclo inhibitors of potassium channel function Bristol-Myers Squibb Company (US) 2011-10-05 EP disclosed
US-20090312307-A1 HETEROCYCLO INHIBITORS OF POTASSIUM CHANNEL FUNCTION BRISTOL-MYERS SQUIBB COMPANY 2009-12-17 US disclosed
US-20090312307-A1 HETEROCYCLO INHIBITORS OF POTASSIUM CHANNEL FUNCTION BRISTOL-MYERS SQUIBB COMPANY 2009-12-17 US disclosed
US-7582654-B2 Heterocyclo inhibitors of potassium channel function BRISTOL-MYERS SQUIBB COMPANY (US) 2009-09-01 US disclosed
US-7582654-B2 Heterocyclo inhibitors of potassium channel function BRISTOL-MYERS SQUIBB COMPANY (US) 2009-09-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090312307-A1 HETEROCYCLO INHIBITORS OF POTASSIUM CHANNEL FUNCTION KCNJ2, KCNH2, KCNQ5 MEN1 3501/4885KMT2A 957/4885GAA 3999/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.