SCHEMBL24723912

SCHEMBL24723912

C=C(OCC)c1cnn(COCC[Si](C)(C)C)c(=O)c1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 2/20 0.35
NPC1 O15118 1/20 0.34
PDE1B Q01064 1/20 0.33
F2RL1 P55085 1/20 0.32
KLKB1 P03952 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2965865 0.86 CYP2C9 (0.42) DGAT1NPC1
SCHEMBL26915876 0.85 NPC1 (0.36) DGAT1NPC1F2RL1KLKB1
SCHEMBL24723914 0.81 NPC1 (0.41) DGAT1NPC1F2RL1KLKB1
SCHEMBL2965634 0.78 NPC1 (0.39) DGAT1NPC1F2RL1KLKB1
SCHEMBL26915819 0.75 F2RL1 (0.33) DGAT1NPC1F2RL1
SCHEMBL18339054 0.75 NPC1 (0.33) DGAT1NPC1F2RL1
SCHEMBL17582616 0.74 PDE1B (0.38) PDE1B
SCHEMBL17582596 0.74 PTGS1 (0.48) PDE1B
SCHEMBL25017777 0.74 CYP2C9 (0.42) NPC1
SCHEMBL26915678 0.73 DGAT1 (0.34) DGAT1NPC1F2RL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240287070-A1 FUSED HETEROCYCLIC DERIVATIVES JOHNSON & JOHNSON (CHINA) INVESTMENT LTD. (CN) 2024-08-29 US disclosed
EP-4347590-A1 FUSED HETEROCYCLIC DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2024-04-10 EP disclosed
CN-117715909-A Condensed heterocyclic derivative 杨森科学爱尔兰无限公司 2024-03-15 CN disclosed
WO-2022253259-A1 FUSED HETEROCYCLIC DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2022-12-08 WO disclosed
WO-2022253259-A1 FUSED HETEROCYCLIC DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2022-12-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240287070-A1 FUSED HETEROCYCLIC DERIVATIVES HAVCR2, HCCS, GOT2 DGAT1 3312/4885NPC1 95/4885PDE1B 4800/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.