SCHEMBL2472745

SCHEMBL2472745

O=P(O)(O)Oc1ccccc1Br

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
INPPL1 O15357 11/20 0.57
INPP5A Q14642 6/20 0.57
INPP5B P32019 2/20 0.57
SRC P12931 4/20 0.55
KDM4E B2RXH2 1/20 0.55
USP2 O75604 1/20 0.55
ALDH1A1 P00352 1/20 0.55
HPGD P15428 1/20 0.55
PDE3A Q14432 1/20 0.55
HSD17B10 Q99714 1/20 0.55
AKT1 P31749 1/20 0.50
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
GRM4 Q14833 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31095030 1.00 INPPL1 (0.57) INPPL1INPP5AINPP5BSRCKDM4E
SCHEMBL2470674 0.87 GPR84 (0.44) INPPL1INPP5AINPP5BSRCKDM4E
Tromethamine SCHEMBL5906711 0.85 INPPL1 (0.43) INPPL1INPP5AINPP5BSRCKDM4E
SCHEMBL2573126 0.84 INPPL1 (0.70) INPPL1INPP5AINPP5BSRCKDM4E
SCHEMBL8054913 0.83 INPPL1 (0.59) INPPL1INPP5AINPP5BSRCKDM4E
SCHEMBL28074624 0.83 HPGD (0.41) INPPL1INPP5AINPP5BSRCKDM4E
SCHEMBL9058386 0.83 INPPL1 (0.39) INPPL1INPP5AINPP5BSRCKDM4E
SCHEMBL29735537 0.82 HTR7 (0.38) INPPL1INPP5AINPP5BSRCKDM4E
SCHEMBL2472741 0.82 HTR7 (0.38) INPPL1INPP5AINPP5BSRCKDM4E
SCHEMBL9765448 0.82 INPPL1 (0.38) INPPL1INPP5AINPP5BSRCKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 59 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006542-A None JP disclosed
WO-2025076861-A1 CARBAZOLE ORGANIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 天合光能股份有限公司 2025-04-17 WO disclosed
CN-117417287-A Carbazole organic compound, and preparation method and application thereof 天合光能股份有限公司 2024-01-19 CN disclosed
US-20230176481-A1 FILM-FORMING COMPOSITION NISSAN CHEMICAL CORPORATION (JP) 2023-06-08 US disclosed
CN-115702149-A Pesticidally active heterocyclic derivatives with sulfur-containing substituents 先正达农作物保护股份公司 2023-02-14 CN disclosed
CN-115697063-A Fungicidal compositions 先正达农作物保护股份公司 2023-02-03 CN disclosed
CN-115398342-A Film-forming composition 日产化学株式会社 2022-11-25 CN disclosed
CN-112105264-B Polymeric dispersants for pesticides 禾大国际股份公开有限公司 2022-08-26 CN disclosed
CN-114814013-A Method for rapidly screening unknown chemical hazard residues in aquatic products based on high-resolution mass spectrum database 中国海洋大学 2022-07-29 CN disclosed
CN-114401963-A Pesticidally active cyclic amine compounds 先正达农作物保护股份公司 2022-04-26 CN disclosed
CN-1314909-A Aryl phosphate derivatives of d4T having anti-HIV activity PARKER HUGHES INST (US) 2001-09-26 CN disclosed
EP-1090018-A1 ARYL PHOSPHATE DERIVATIVES OF d4T HAVING ANTI-HIV ACTIVITY Parker Hughes Institute (US) 2001-04-11 EP disclosed
US-6140508-A USEFUL IN THE PREPARATION OF FARNESYL-PROTEIN TRANSFERASE INHIBITORS. MERCK & CO., INC. (US) 2000-10-31 US disclosed
US-6030957-A INHIBITING HIV(HUMAN IMMUNODEFICIENCY VIRUS) REVERSE TRANSCIPTASE IN CELLS INFECTED WITH HIV BY ADMINISTERING TO INFECTED CELLS ARYLPHOSPHATE DERIVATIVE OF 2',3'-DIDEHYDRO-2',3'-DIDEOXYTHYMIDINE WAYNE HUGHES INSTITUTE (US) 2000-02-29 US disclosed
WO-2000001691-A1 PROCESS FOR MAKING FARNESYL-PROTEIN TRANSFERASE INHIBITORS MERCK & CO., INC. (US) 2000-01-13 WO disclosed
WO-2000001674-A1 PROCESS FOR MAKING 1,5-DISUBSTITUTED IMIDAZOLES MERCK & CO., INC. (US) 2000-01-13 WO disclosed
WO-2000000501-A1 ARYL PHOSPHATE DERIVATIVES OF d4T HAVING ANTI-HIV ACTIVITY PARKER HUGHES INSTITUTE (US) 2000-01-06 WO disclosed
CN-1067247-A The method of purifying polybrominated triaryl phosphate esters FMC CORP (US) 1992-12-23 CN disclosed
US-4992496-A Polybrominated aryl phosphate ester and epoxy compound FMC CORPORATION (US) 1991-02-12 US disclosed
JP-H026542-A FLAME-RETARDANT THERMOPLASTIC COMPOSITION COMPRISING POLYBROMOPHENYL PHOSPHATE FMC CORP 1990-01-10 JP disclosed