SCHEMBL24735339

SCHEMBL24735339

Nc1ccc(N2CCC(CO)C2)c(F)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
LMNA P02545 1/20 0.48
MAPT P10636 1/20 0.48
MAPK1 P28482 1/20 0.48
GFER P55789 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
SYK P43405 2/20 0.39
HTT P42858 2/20 0.39
BPTF Q12830 1/20 0.39
GAA P10253 3/20 0.39
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NOTUM Q6P988 1/20 0.37
LPL P06858 1/20 0.37
LIPG Q9Y5X9 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
CDK8 P49336 1/20 0.36
SLC6A9 P48067 1/20 0.36
GPR55 Q9Y2T6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24735594 1.00 ALDH1A1 (0.48) ALDH1A1LMNAMAPTMAPK1GFER
SCHEMBL24735237 1.00 ALDH1A1 (0.48) ALDH1A1LMNAMAPTMAPK1GFER
SCHEMBL9983818 0.92 ALDH1A1 (0.46) ALDH1A1LMNAMAPTMAPK1GFER
SCHEMBL20231853 0.91 MAPT (0.54) ALDH1A1LMNAMAPTMAPK1GFER
SCHEMBL29890862 0.91 MAPT (0.54) ALDH1A1LMNAMAPTMAPK1GFER
SCHEMBL24735187 0.88 ALDH1A1 (0.49) ALDH1A1LMNAMAPTMAPK1GFER
SCHEMBL5201699 0.84 ALDH1A1 (0.44) ALDH1A1LMNAMAPTMAPK1GFER
SCHEMBL5201691 0.84 ALDH1A1 (0.44) ALDH1A1LMNAMAPTMAPK1GFER
SCHEMBL24735592 0.83 SYK (0.39) MAPTSYKBPTFGAAHPGD
SCHEMBL24735234 0.83 SYK (0.39) MAPTSYKBPTFGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117042769-A Substituted pyrrolopyrimidines and pyrazolopyrimidines as Bruton's Tyrosine Kinase (BTK) degrading agents 冰洲石生物科技公司 2023-11-10 CN disclosed
US-11530222-B2 Substituted pyrrolopyrimidine and pyrazolopyrimidine as Bruton's tyrosine kinase (BTK) degraders ACCUTAR BIOTECHNOLOGY INC. (US) 2022-12-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11530222-B2 Substituted pyrrolopyrimidine and pyrazolopyrimidine as Bruton's tyrosine kinase (BTK) degraders BTK, LYN, SYK ALDH1A1 2925/4885LMNA 4497/4885MAPT 4299/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.