SCHEMBL24740459

SCHEMBL24740459

O=C(O)CC[C@H]1CCCN1c1cc(C(F)(F)F)c(OCc2ccccc2)nn1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TIPARP Q7Z3E1 2/20 0.42
TACR1 P25103 2/20 0.37
SPHK2 Q9NRA0 3/20 0.37
ITGB2 P05107 3/20 0.37
ICAM1 P05362 3/20 0.37
ITGAL P20701 3/20 0.37
AADAT Q8N5Z0 1/20 0.37
SPHK1 Q9NYA1 3/20 0.36
FFAR1 O14842 1/20 0.36
CHRNB2 P17787 2/20 0.36
CHRNA7 P36544 2/20 0.36
CHRNA4 P43681 2/20 0.36
CHRNA5 P30532 1/20 0.36
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35
S1PR1 P21453 1/20 0.35
IDH1 O75874 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24739046 1.00 TIPARP (0.42) TIPARPTACR1SPHK2ITGB2ICAM1
SCHEMBL24739045 0.90 POLB (0.39) TIPARPITGB2ICAM1ITGALCHRNB2
SCHEMBL24740461 0.90 POLB (0.39) TIPARPITGB2ICAM1ITGALCHRNB2
SCHEMBL24740462 0.86 TIPARP (0.64) TIPARP
SCHEMBL24739041 0.86 TIPARP (0.64) TIPARP
SCHEMBL24740409 0.85 THRA (0.35) FFAR1RXRARXRBRXRGS1PR1
SCHEMBL24739382 0.81 FFAR1 (0.35) FFAR1RXRARXRBRXRGS1PR1
SCHEMBL24739385 0.80 TIPARP (0.54) TIPARPAADAT
SCHEMBL28914953 0.79 TIPARP (0.46) TIPARPTACR1FFAR1
SCHEMBL28914956 0.79 TIPARP (0.46) TIPARPTACR1FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022253101-A1 PYRIDAZINONE COMPOUND AS PARP7 INHIBITOR 上海优理惠生医药有限公司 2022-12-08 WO disclosed