SCHEMBL24744334

SCHEMBL24744334

COC(=O)c1cc2c([nH]1)-c1ccccc1CC2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.51
KDM4E B2RXH2 5/20 0.51
HPGD P15428 4/20 0.51
L3MBTL1 Q9Y468 3/20 0.51
XDH P47989 1/20 0.43
LMNA P02545 1/20 0.42
NOTUM Q6P988 1/20 0.42
SRD5A1 P18405 1/20 0.42
SRD5A2 P31213 1/20 0.42
GAA P10253 4/20 0.41
RAB9A P51151 3/20 0.41
NPC1 O15118 2/20 0.41
CYP1A2 P05177 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
MAPT P10636 2/20 0.40
TSHR P16473 2/20 0.40
TDP1 Q9NUW8 1/20 0.39
BRD4 O60885 1/20 0.39
GLA P06280 2/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30115707 0.83 SRD5A2 (0.51) ALDH1A1KDM4EHPGDLMNANOTUM
SCHEMBL3607213 0.81 CCNC (0.53) ALDH1A1KDM4EGAACYP1A2GLA
SCHEMBL1005097 0.78 CYP1A2 (0.49) KDM4EL3MBTL1XDHLMNASRD5A1
SCHEMBL1005747 0.78 MIF (0.45) ALDH1A1L3MBTL1XDHLMNAGAA
SCHEMBL1005746 0.78 MIF (0.45) ALDH1A1L3MBTL1XDHLMNAGAA
SCHEMBL31062548 0.77 MAPT (0.37) ALDH1A1KDM4EHPGDL3MBTL1LMNA
SCHEMBL24746391 0.73 HPGD (0.45) ALDH1A1KDM4EHPGDL3MBTL1LMNA
SCHEMBL24744751 0.73 CCNC (0.44) ALDH1A1KDM4EHPGDL3MBTL1LMNA
SCHEMBL24746390 0.72 KDM4E (0.44) ALDH1A1KDM4EHPGDL3MBTL1LMNA
SCHEMBL21356990 0.72 KDM4E (0.50) ALDH1A1KDM4EHPGDLMNANOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4347595-A1 SUBSTITUTED TRICYCLIC HETEROCYCLIC COMPOUNDS AS METALLO-BETA-LACTAMASE INHIBITORS Council of Scientific & Industrial Research (IN) 2024-04-10 EP disclosed
WO-2022254464-A1 SUBSTITUTED TRICYCLIC HETEROCYCLIC COMPOUNDS AS METALLO-BETA-LACTAMASE INHIBITORS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2022-12-08 WO disclosed
WO-2022254464-A1 SUBSTITUTED TRICYCLIC HETEROCYCLIC COMPOUNDS AS METALLO-BETA-LACTAMASE INHIBITORS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2022-12-08 WO disclosed