SCHEMBL24745882

SCHEMBL24745882

CC1(O)CCN(c2ccc(Nc3cc(Cl)nc4cc[nH]c(=O)c34)nc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SYK P43405 5/20 0.43
MAP4K1 Q92918 3/20 0.39
CDK4 P11802 3/20 0.39
TYK2 P29597 4/20 0.38
JAK2 O60674 4/20 0.38
CDK6 Q00534 1/20 0.36
EGFR P00533 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29891033 1.00 SYK (0.43) SYKMAP4K1CDK4TYK2JAK2
SCHEMBL24745826 0.87 TYK2 (0.47) MAP4K1CDK4TYK2
SCHEMBL29891142 0.87 TYK2 (0.47) MAP4K1CDK4TYK2
SCHEMBL610905 0.76 SYK (0.43) SYKMAP4K1CDK4TYK2JAK2
SCHEMBL24747223 0.76 TYK2 (0.46) MAP4K1CDK4TYK2
SCHEMBL24745891 0.76 TYK2 (0.46) SYKMAP4K1CDK4TYK2
SCHEMBL29891207 0.76 TYK2 (0.46) SYKMAP4K1CDK4TYK2
SCHEMBL30316297 0.76 TYK2 (0.46) MAP4K1CDK4TYK2
SCHEMBL24745833 0.75 MAP4K1 (0.47) MAP4K1CDK4CDK6EGFR
SCHEMBL24746072 0.75 CDK4 (0.45) CDK4CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117120090-A HPK1 antagonists and uses thereof 林伯士萨顿公司 2023-11-24 CN disclosed
WO-2022174253-A1 HPK1 ANTAGONISTS AND USES THEREOF Nimbus Saturn, Inc. (US) 2022-08-18 WO disclosed