SCHEMBL24765638

SCHEMBL24765638

COc1cc(Sc2ccccc2)c(OC)cc1C=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.53
TDP1 Q9NUW8 2/20 0.53
KDM4E B2RXH2 2/20 0.53
TSHR P16473 1/20 0.53
PRKDC P78527 2/20 0.45
MAPT P10636 4/20 0.43
HPGD P15428 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
ALOX15 P16050 2/20 0.43
HSD17B10 Q99714 2/20 0.43
GAA P10253 1/20 0.43
MAPK1 P28482 1/20 0.43
FGFR1 P11362 1/20 0.43
LMNA P02545 3/20 0.41
NPC1 O15118 1/20 0.40
POLB P06746 1/20 0.40
RAB9A P51151 1/20 0.40
ERN1 O75460 4/20 0.39
TLR2 O60603 1/20 0.39
TLR1 Q15399 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9954218 0.89 ALDH1A1 (0.50) ALDH1A1TDP1KDM4ETSHRPRKDC
SCHEMBL10486972 0.78 TTR (0.55) ALDH1A1TDP1TSHRMAPTHPGD
SCHEMBL5113878 0.78 TTR (0.55) ALDH1A1TDP1TSHRMAPTHPGD
SCHEMBL27135190 0.77 FBP1 (0.44) ALDH1A1TDP1MAPTHPGDL3MBTL1
SCHEMBL27002062 0.77 FBP1 (0.44) ALDH1A1TDP1MAPTHPGDL3MBTL1
SCHEMBL11615151 0.76 ALDH1A1 (0.64) ALDH1A1TDP1KDM4ETSHRPRKDC
SCHEMBL29965864 0.76 MAPT (0.38) ALDH1A1TDP1KDM4EMAPTHPGD
SCHEMBL3136850 0.75 ALDH1A1 (0.90) ALDH1A1TDP1KDM4ETSHRPRKDC
SCHEMBL16495093 0.75 ERN1 (0.50) ALDH1A1TDP1KDM4EMAPTLMNA
SCHEMBL3848297 0.74 KMT2A (0.44) ALDH1A1TDP1KDM4ETSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117642379-A Phenylalkylamines and methods of making and using the same 吉尔伽美什制药公司 2024-03-01 CN disclosed
WO-2022204323-A1 NON-HALLUCINOGENIC ARIADNE ANALOGS FOR TREATMENT OF NEUROLOGICAL AND PSYCHIATRIC DISORDERS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2022-09-29 WO disclosed