SCHEMBL24769722

SCHEMBL24769722

COc1cnc(Cl)cc1-c1cc(F)ccc1C(C)=O

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 1/20 0.43
KCNQ2 O43526 1/20 0.43
POLQ O75417 11/20 0.42
GPBAR1 Q8TDU6 1/20 0.40
PDE10A Q9Y233 1/20 0.38
DHFR P00374 1/20 0.38
DHODH Q02127 1/20 0.38
CSF1R P07333 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24769729 0.83 SMN1; SMN2 (0.43) POLQDHFR
SCHEMBL24770364 0.81 POLQ (0.44) KCNQ3KCNQ2POLQDHFR
SCHEMBL24769992 0.78 POLQ (0.70) POLQ
SCHEMBL19945811 0.75 MEN1 (0.47)
SCHEMBL29479275 0.75 MEN1 (0.47)
SCHEMBL29276870 0.73 POLQ (0.44) POLQ
SCHEMBL16368532 0.73 HTT (0.46) KCNQ3KCNQ2POLQPDE10A
SCHEMBL31248788 0.73 HTT (0.46) KCNQ3KCNQ2POLQPDE10A
SCHEMBL31541641 0.72 POLQ (0.43) POLQDHFR
SCHEMBL19945742 0.72 ALDH1A1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022259204-A1 O-LINKED THIADIAZOLYL COMPOUNDS AS DNA POLYMERASE THETA INHIBITORS IDEAYA BIOSCIENCES, INC. (US) 2022-12-15 WO disclosed