SCHEMBL24770276

SCHEMBL24770276

COC(=O)/C(N)=C(O)/C=C(/C)N

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
EGLN1 Q9GZT9 1/20 0.30
OPRK1 P41145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24770338 0.77 ALDH1A1 (0.34) ALDH1A1
SCHEMBL21503761 0.74
SCHEMBL18714044 0.72
SCHEMBL25156142 0.71 ALDH1A1 (0.48) ALDH1A1MAPTEGLN1OPRK1
SCHEMBL2246387 0.71
SCHEMBL19366418 0.71
SCHEMBL822962 0.69
SCHEMBL62213 0.69
SCHEMBL62212 0.69
SCHEMBL23369533 0.69 ALDH1A1 (0.38) ALDH1A1EGLN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022259204-A1 O-LINKED THIADIAZOLYL COMPOUNDS AS DNA POLYMERASE THETA INHIBITORS IDEAYA BIOSCIENCES, INC. (US) 2022-12-15 WO disclosed