SCHEMBL2477950

SCHEMBL2477950

C=CCC(N)c1ccccc1-c1cc(Cl)ccc1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1LG2 Q9BQ51 2/20 0.41
CD274 Q9NZQ7 2/20 0.41
PLA2G7 Q13093 1/20 0.37
SCN4A P35499 4/20 0.36
S100A4 P26447 1/20 0.34
CHRM1 P11229 1/20 0.34
CYP3A4 P08684 1/20 0.33
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CASP3 P42574 1/20 0.32
RAB9A P51151 1/20 0.32
SENP8 Q96LD8 1/20 0.32
SENP7 Q9BQF6 1/20 0.32
SENP6 Q9GZR1 1/20 0.32
ATM Q13315 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
IDO1 P14902 1/20 0.32
DPP4 P27487 1/20 0.32
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2473732 0.84 PDCD1LG2 (0.36) PDCD1LG2CD274PLA2G7CYP3A4
SCHEMBL2476189 0.81 PDCD1LG2 (0.39) PDCD1LG2CD274S100A4ATML3MBTL1
SCHEMBL2473298 0.78 PDCD1LG2 (0.44) PDCD1LG2CD274PLA2G7CYP3A4NPC1
SCHEMBL2474146 0.78 PDCD1LG2 (0.45) PDCD1LG2CD274CYP3A4ALDH1A1CASP3
SCHEMBL8995483 0.77 ESR1 (0.41) PDCD1LG2CD274SCN4ACHRM1CYP3A4
SCHEMBL2474504 0.75 ALOX5AP (0.38) PDCD1LG2CD274DPP4TP53
SCHEMBL2474346 0.73 PDCD1LG2 (0.36) PDCD1LG2CD274
SCHEMBL6712688 0.73 ESR1 (0.38) PDCD1LG2CD274ALDH1A1
SCHEMBL6712687 0.73 ESR1 (0.38) PDCD1LG2CD274ALDH1A1
Hydrochloric Acid SCHEMBL2476355 0.73 PDCD1LG2 (0.37) PDCD1LG2CD274KDM4ENPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2159216-B1 3-BUTENYL-1-AMINE DERIVATIVES AND THEIR USE AS Ih MODULORS FOR THE TREATMENT OF PSYCHIATIRC DISORDERS ORGANON NV (NL) 2011-10-12 EP disclosed
EP-2159216-A1 Ih - Modulators N.V. Organon (NL) 2010-03-03 EP disclosed
US-20020037885-A1 Therapeutic compounds DIJCKS FREDERICUS ANTONIUS (NL) 2002-03-28 US disclosed
US-6313139-B1 ADMINISTERING BENZYLAMINE DERIVATIVE FOR THERAPY OF PSYCHIATRIC DISORDER IN MAMMALS AKZO NOBEL N. V. (NL) 2001-11-06 US disclosed
EP-1035843-A2 I h?-MODULATORS Akzo Nobel N.V. (NL) 2000-09-20 EP disclosed
US-6080773-A USEFUL FOR TREATMENT OF DEPRESSION, ANXIETY OR PSYCHOSIS AKZO NOBEL, N.V. (NL) 2000-06-27 US disclosed
WO-1999018941-A2 Ih-MODULATORS AKZO NOBEL N.V. (NL) 1999-04-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020037885-A1 Therapeutic compounds BDNF, PNMT, SLC18A2 PDCD1LG2 3624/4885CD274 2894/4885PLA2G7 2175/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.