SCHEMBL24780883

SCHEMBL24780883

CNc1cc2ccc(Br)cc2s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 3/20 0.43
RAB9A P51151 3/20 0.37
DYRK1A Q13627 2/20 0.37
NPC1 O15118 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
CYP2A6 P11509 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28469540 0.85 HSP90AA1 (0.47) APPRAB9ADYRK1ANPC1CYP1A2
SCHEMBL25809470 0.78 HDAC3 (0.50) APPRAB9ADYRK1ANPC1CYP1A2
SCHEMBL6813386 0.74 APP (0.41) APPRAB9ADYRK1ANPC1CYP1A2
SCHEMBL31009687 0.74 CYP2A6 (0.38) APPRAB9ADYRK1ANPC1CYP1A2
SCHEMBL3962610 0.74 CYP2A6 (0.38) APPRAB9ADYRK1ANPC1CYP1A2
SCHEMBL18878582 0.73 CYP2A6 (0.41) APPRAB9ADYRK1ANPC1CYP1A2
SCHEMBL21234680 0.72 CYP2A6 (0.34) RAB9ADYRK1ANPC1CYP2A6ALDH1A1
SCHEMBL6121215 0.71 CYP2A6 (0.39) APPRAB9ADYRK1ANPC1CYP1A2
SCHEMBL24780599 0.71 RAB9A (0.44) RAB9ADYRK1ANPC1CYP1A2CYP3A4
SCHEMBL3478461 0.71 RAB9A (0.40) APPRAB9ADYRK1ANPC1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118894816-A 3, 3-Difluoroallylamine or salt thereof and pharmaceutical composition comprising the same 柳韩洋行 2024-11-05 CN disclosed
CN-113330001-B 3, 3-Difluoroallylamine or salt thereof and pharmaceutical composition comprising the same 柳韩洋行 2024-07-02 CN disclosed
WO-2022263557-A1 PHARMACEUTICAL COMPOUND GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2022-12-22 WO disclosed
CN-113330001-A 3, 3-difluoroallylamine or salt thereof and pharmaceutical composition containing same 柳韩洋行 2021-08-31 CN disclosed