SCHEMBL3478461

SCHEMBL3478461

COc1cc2ccc(Br)cc2s1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.40
CA2 P00918 1/20 0.37
XPO1 O14980 1/20 0.36
CYP2A6 P11509 1/20 0.35
NPC1 O15118 2/20 0.35
MGAM O43451 1/20 0.35
GAA P10253 1/20 0.35
SI P14410 1/20 0.35
MGAM2 Q2M2H8 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
DYRK1A Q13627 1/20 0.35
HDAC1 Q13547 1/20 0.35
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35
TUBA3C P0DPH7 1/20 0.35
TUBA1B P68363 1/20 0.35
TUBA4A P68366 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3478352 0.84 HSP90AA1 (0.49) RAB9ACA2XPO1CYP2A6MGAM
SCHEMBL5201465 0.78 RAB9A (0.46) RAB9ANPC1CYP1A2CYP3A4CYP2C9
SCHEMBL29239834 0.78 CA2 (0.57) RAB9ACA2CYP2A6NPC1CYP1A2
SCHEMBL3962610 0.75 CYP2A6 (0.38) RAB9ACYP2A6NPC1CYP1A2CYP3A4
SCHEMBL31009687 0.75 CYP2A6 (0.38) RAB9ACYP2A6NPC1CYP1A2CYP3A4
SCHEMBL18950282 0.74 CA2 (0.40) RAB9ACA2CYP2A6NPC1CYP1A2
SCHEMBL14761513 0.74 RAB9A (0.36) RAB9ACA2CYP2A6NPC1CYP1A2
SCHEMBL5202024 0.74 RAB9A (0.39) RAB9ANPC1CYP1A2CYP3A4CYP2C9
SCHEMBL18878582 0.74 CYP2A6 (0.41) RAB9ACYP2A6NPC1CYP1A2CYP3A4
SCHEMBL147625 0.72 TUBB4A (0.46) CA2CYP2A6CYP1A2HDAC1TUBB4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2167083-A2 NOVEL 1- HETEROARYL-3-AZABICYCLOÝ3.1.0¨HEXANES, METHODS FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS DOV Pharmaceutical, Inc. (US) 2010-03-31 EP disclosed
WO-2008153937-A2 NOVEL 1- HETEROARYL-3-AZABICYCLO[3.1.0]HEXANES, METHODS FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS DOV PHARMACEUTICAL, INC. (US) 2008-12-18 WO disclosed